Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50022260
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649929(CHEMBL5630432)
Affinity DataIC50: 250nMAssay Description:Inhibition of PKM2 (unknown origin) by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649932(CHEMBL5630549)
Affinity DataIC50: 303nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649929(CHEMBL5630432)
Affinity DataIC50: 350nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649946(CHEMBL5624918)
Affinity DataIC50: 362nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649935(CHEMBL5624981)
Affinity DataIC50: 380nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649945(CHEMBL5624442)
Affinity DataIC50: 420nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649929(CHEMBL5630432)
Affinity DataIC50: 477nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649933(CHEMBL5630450)
Affinity DataIC50: 478nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649935(CHEMBL5624981)
Affinity DataIC50: 517nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649946(CHEMBL5624918)
Affinity DataIC50: 542nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649932(CHEMBL5630549)
Affinity DataIC50: 545nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649945(CHEMBL5624442)
Affinity DataIC50: 572nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649936(CHEMBL5624782)
Affinity DataIC50: 572nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649934(CHEMBL5630893)
Affinity DataIC50: 603nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649933(CHEMBL5630450)
Affinity DataIC50: 610nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649936(CHEMBL5624782)
Affinity DataIC50: 637nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649934(CHEMBL5630893)
Affinity DataIC50: 854nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649939(CHEMBL5624871)
Affinity DataIC50: 897nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649948(CHEMBL5630822)
Affinity DataIC50: 901nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649938(CHEMBL5630750)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649937(CHEMBL5625056)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649944(CHEMBL5624978)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649943(CHEMBL5631103)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649941(CHEMBL5631060)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649947(CHEMBL5630212)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649942(CHEMBL5624534)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649940(CHEMBL5630214)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649931(CHEMBL5630287)
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649931(CHEMBL5630287)
Affinity DataIC50: 2.92E+3nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649930(CHEMBL5624751)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM7458(Naringenin, 18 | 5,7-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin) in presence of FBP by Michaelis-menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM7458(Naringenin, 18 | 5,7-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)TBA
LigandPNGBDBM50649930(CHEMBL5624751)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal his8-tagged PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed