Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50022284
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650275(CHEMBL5631076)
Affinity DataIC50: 5.90nMAssay Description:Inverse agonist activity at human N-terminal his 6 tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) cells incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50512497(CHEMBL4567440)
Affinity DataIC50: 44nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) incubated for 15 mins by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650279(CHEMBL5629900)
Affinity DataIC50: 50nMAssay Description:Inhibition of RORgamma (unknown origin) incubated for 1 hr by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650278(CHEMBL5630956)
Affinity DataIC50: 50nMAssay Description:Inhibition of RORgamma (unknown origin) incubated for 1 hr by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650277(CHEMBL5630700)
Affinity DataIC50: 50nMAssay Description:Inhibition of RORgamma (unknown origin) incubated for 1 hr by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650276(CHEMBL5630221)
Affinity DataIC50: 50nMAssay Description:Inhibition of RORgamma (unknown origin) incubated for 1 hr by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650283(CHEMBL5629952)
Affinity DataIC50: 50nMAssay Description:Inhibition of RORgamma (unknown origin) incubated for 1 hr by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650282(CHEMBL5629926)
Affinity DataIC50: 50nMAssay Description:Inhibition of RORgamma (unknown origin) incubated for 1 hr by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650281(CHEMBL5630789)
Affinity DataIC50: 50nMAssay Description:Inhibition of RORgamma (unknown origin) incubated for 1 hr by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650280(CHEMBL5624671)
Affinity DataIC50: 50nMAssay Description:Inhibition of RORgamma (unknown origin) incubated for 1 hr by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50106301(CHEMBL3598140)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataEC50:  340nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50519881(CHEMBL4435145)
Affinity DataIC50: 425nMAssay Description:Inhibition of RORgamma (unknown origin) incubated for 1 hr by TR-FRET methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50103521(CHEBI:8228 | Actos | Duetact | Pioglitazone | US20...)
Affinity DataEC50:  720nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor ROR-alpha(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650275(CHEMBL5631076)
Affinity DataIC50: 4.00E+3nMAssay Description:Inverse agonist activity at human his 6 tagged RORalpha LBD incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50650275(CHEMBL5631076)
Affinity DataIC50: 1.00E+5nMAssay Description:Inverse agonist activity at human his 6 tagged PPARgammaLBD incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed