Compile Data Set for Download or QSAR
Report error Found 220 Enz. Inhib. hit(s) with all data for entry = 50019395
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424409BDBM424409(US10508120, Compound I-922 | US10508120, Compound ...)
Affinity DataKd:  0.00100nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424440BDBM424440(US10508120, Compound I-1074 | US10508120, Compound...)
Affinity DataKd:  0.00100nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 565685BDBM565685(US11414431, Compound I-253 | US12221453, Compound ...)
Affinity DataKd:  0.00200nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424362BDBM424362(US10508120, Compound I-817 | US10508120, Compound ...)
Affinity DataKd:  0.00200nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 565687BDBM565687(US11414431, Compound I-255 | US12221453, Compound ...)
Affinity DataKd:  0.00200nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424815BDBM424815(US10508120, Compound I-1319 | US10577373, Compound...)
Affinity DataKd:  0.00200nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424435BDBM424435(US10508120, Compound I-975 | US10508120, Compound ...)
Affinity DataKd:  0.00200nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424662BDBM424662(US10508120, Compound I-1117 | US10577373, Compound...)
Affinity DataKd:  0.00300nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424408BDBM424408(US10508120, Compound I-904 | US10508120, Compound ...)
Affinity DataKd:  0.00300nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424408BDBM424408(US10508120, Compound I-904 | US10508120, Compound ...)
Affinity DataKd:  0.00300nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424448BDBM424448(US10508120, Compound I-903 | US10577373, Compound ...)
Affinity DataKd:  0.00400nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618789BDBM50618789(CHEMBL5438635)
Affinity DataKd:  0.00400nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424559BDBM424559(US10508120, Compound I-1353 | US10508120, Compound...)
Affinity DataKd:  0.00400nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424454BDBM424454(US10508120, Compound I-1183 | US10508120, Compound...)
Affinity DataKd:  0.00400nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424525BDBM424525(US10508120, Compound I-980 | US10577373, Compound ...)
Affinity DataKd:  0.00400nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424893BDBM424893(US10508120, Compound I-1397 | US10577373, Compound...)
Affinity DataKd:  0.00500nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424422BDBM424422(US10508120, Compound I-877 | US10577373, Compound ...)
Affinity DataKd:  0.00600nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 565683BDBM565683(US11414431, Compound I-251 | US12221453, Compound ...)
Affinity DataKd:  0.00600nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424529BDBM424529(US10508120, Compound I-1084 | US10508120, Compound...)
Affinity DataKd:  0.00600nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424220BDBM424220(US10508120, Compound I-675 | US10508120, Compound ...)
Affinity DataKd:  0.00700nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 565754BDBM565754(US11414431, Compound I-322 | US12221453, Compound ...)
Affinity DataKd:  0.00800nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424111BDBM424111(US10508120, Compound I-572 | US10577373, Compound ...)
Affinity DataKd:  0.0190nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424808BDBM424808(US10508120, Compound I-1413 | US10508120, Compound...)
Affinity DataKd:  0.0230nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424086BDBM424086(US10577373, Compound I-541 | US10508120, Compound ...)
Affinity DataKd:  0.0330nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424388BDBM424388(US10508120, Compound I-973 | US10508120, Compound ...)
Affinity DataKd:  0.0340nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 423553BDBM423553(US10508120, Compound I-175 | US10508120, Compound ...)
Affinity DataKd:  0.0390nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 423652BDBM423652(US10508120, Compound I-107 | US10577373, Compound ...)
Affinity DataKd:  0.0630nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [5-1181](Mouse)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424454BDBM424454(US10508120, Compound I-1183 | US10508120, Compound...)
Affinity DataKd:  0.0670nMAssay Description:Binding affinity to mouse TYK2 JH2 domain assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 435794BDBM435794(US10577373, Compound I-954)
Affinity DataKd:  0.0680nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 423689BDBM423689(US10508120, Compound I-144 | US10577373, Compound ...)
Affinity DataKd:  0.0730nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 423409BDBM423409(US10508120, Compound I-1 | US10577373, Compound I-...)
Affinity DataKd:  0.0780nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 565847BDBM565847(US11414431, Compound I-415 | US12221453, Compound ...)
Affinity DataKd:  0.0860nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50526606BDBM50526606(CHEMBL4532948 | US11174264, Compound I-3)
Affinity DataKi:  0.0860nMAssay Description:Inhibition of TYK2 JH2 domain (unknown origin) in presence of 10 uM of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424807BDBM424807(US10508120, Compound I-1311 | US10577373, Compound...)
Affinity DataKd:  0.0880nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 423688BDBM423688(US10508120, Compound I-143 | US10577373, Compound ...)
Affinity DataKd:  0.0990nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424410BDBM424410(US10508120, Compound I-924 | US10508120, Compound ...)
Affinity DataKd:  0.105nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424321BDBM424321(US10508120, Compound I-776 | US10577373, Compound ...)
Affinity DataKd:  0.130nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50526603BDBM50526603(CHEMBL4293907)
Affinity DataKi:  0.130nMAssay Description:Inhibition of TYK2 JH2 domain (unknown origin) in presence of 10 uM of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565967BDBM50565967(CHEMBL4784391)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of TYK2 JH2 domain (unknown origin) by HTRF based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424450BDBM424450(US10508120, Compound I-905 | US10577373, Compound ...)
Affinity DataKd:  0.200nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50507816BDBM50507816(Bms-986165 | Deucravacitinib | US12351572, Example...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of TYK2 JH2 domain (unknown origin) by HTRF based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50618788BDBM50618788(CHEMBL5427213)
Affinity DataKd:  0.310nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50507816BDBM50507816(Bms-986165 | Deucravacitinib | US12351572, Example...)
Affinity DataKd:  0.330nMAssay Description:Binding affinity to human JAK1 JH2 domain assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 565510BDBM565510(US11414431, Compound I-76 | US12221453, Compound I...)
Affinity DataKd:  0.380nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424040BDBM424040(US10577373, Compound I-495 | US10508120, Compound ...)
Affinity DataKd:  0.460nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424118BDBM424118(US10577373, Compound I-573 | US10508120, Compound ...)
Affinity DataKd:  0.480nMAssay Description:Binding affinity to human wild type TYK2 JH2 domain (G556/D888) expressed in mammalian expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 406663BDBM406663(US10336752, Compound 2 | US10336752, Compound 4 | ...)
Affinity DataKi:  0.510nMAssay Description:Inhibition of TYK2 JH1 domain (unknown origin) in presence of 10 uM of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424454BDBM424454(US10508120, Compound I-1183 | US10508120, Compound...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of TYK2 dependent IFNalpha-stimulated STAT3 phosphorylation in human PBMCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424815BDBM424815(US10508120, Compound I-1319 | US10577373, Compound...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of TYK2 in human PBMC cells assessed as IL-12 induced phosphorylation of STAT4 levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Nimbus Therapeutics

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 424435BDBM424435(US10508120, Compound I-975 | US10508120, Compound ...)
Affinity DataIC50: 2nMAssay Description:Inhibition of TYK2 in human PBMC cells assessed as IL-12 induced phosphorylation of STAT4 levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
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