Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50020188
TargetSodium channel protein type 9 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human Nav 1.7 expressed in HEK293T cells assessed as phasic block at 10 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as phasic block at 10 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of human Nav 1.7 expressed in HEK293T cells assessed as phasic block at 10 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of human Nav 1.7 expressed in HEK293T cells assessed as phasic block at 10 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as phasic block at 10 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of human Nav 1.7 expressed in HEK293T cells assessed as tonic block at 0.1 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as phasic block at 10 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibition of human Nav 1.7 expressed in HEK293T cells assessed as tonic block at 0.1 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as tonic block at 0.1 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as phasic block at 10 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as tonic block at 0.1 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as phasic block at 10 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 9.50E+4nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as tonic block at 0.1 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of human Nav 1.7 expressed in HEK293T cells assessed as tonic block at 0.1 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 1.18E+5nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as tonic block at 0.1 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro
Curated by ChEMBL
University of Bari Aldo Moro
Curated by ChEMBL
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of human Nav 1.4 expressed in HEK293T cells assessed as tonic block at 0.1 Hz by whole cell patch clamp assayMore data for this Ligand-Target Pair


3D Structure (crystal)

