Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50020263
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50200880(2-hydroxy-N,N-dimethyl-3-{2-[[(R)-1-(5-methylfuran...)
Affinity DataKd:  0.0490nMAssay Description:Displacement of [3H]Sch527123 from human CXCR2 assessed as dissociation constant measured every 30 secs for 48 hrs by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628237(CHEMBL5414239)
Affinity DataKd:  9nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR2 (unknown origin) expressed in HEK293 cell membrane assessed as dissociation constant using furimazine as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628239(CHEMBL5412421)
Affinity DataKd:  27nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR2 (unknown origin) expressed in HEK293 cell membrane assessed as dissociation constant using furimazine as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628238(CHEMBL5413545)
Affinity DataKd:  45nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR2 (unknown origin) expressed in HEK293 cell membrane assessed as dissociation constant using furimazine as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628237(CHEMBL5414239)
Affinity DataKd:  52nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR2 (unknown origin) expressed in HEK293 cells assessed as dissociation constant using furimazine as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628238(CHEMBL5413545)
Affinity DataKd:  82nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR2 (unknown origin) expressed in HEK293 cells assessed as dissociation constant using furimazine as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628239(CHEMBL5412421)
Affinity DataKd:  88nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR2 (unknown origin) expressed in HEK293 cells assessed as dissociation constant using furimazine as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 1(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628237(CHEMBL5414239)
Affinity DataKd:  101nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR1 (unknown origin) expressed in HEK293 cell membrane assessed as dissociation constant using furimazine as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628235(CHEMBL5420355)
Affinity DataKd:  137nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR2 (unknown origin) expressed in HEK293 cell membrane assessed as dissociation constant using furimazine as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628235(CHEMBL5420355)
Affinity DataKd:  149nMAssay Description:Binding affinity to CXCR2 (unknown origin) (28 to 99 residues) expressed in HEK293 cell membrane assessed as dissociation constant using furimazine a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628236(CHEMBL5422785)
Affinity DataKd:  301nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR2 (unknown origin) expressed in HEK293 cell membrane assessed as dissociation constant using furimazine as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 1(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628239(CHEMBL5412421)
Affinity DataKd:  372nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR1 (unknown origin) expressed in HEK293 cell membrane assessed as dissociation constant using furimazine as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetC-X-C chemokine receptor type 2(Human)
University of Nottingham Biodiscovery Institute

Curated by ChEMBL
LigandPNGBDBM50628235(CHEMBL5420355)
Affinity DataKd:  549nMAssay Description:Binding affinity to NanoLuc fused Snap CXCR2 (unknown origin) expressed in HEK293 cells assessed as dissociation constant using furimazine as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed