Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50019307
TargetGuanine nucleotide-binding protein G(i) subunit alpha-1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50617966(CHEMBL5408357)
Affinity DataKd:  710nMAssay Description:Binding affinity to N-terminal 6His-tagged GMPPNP-bound Galphai1 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetGuanine nucleotide-binding protein G(i) subunit alpha-1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50617966(CHEMBL5408357)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to N-terminal 6His-tagged GDP-bound Galphai1 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetGuanine nucleotide-binding protein G(i) subunit alpha-1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50617965(CHEMBL5407838)
Affinity DataKd:  2.47E+4nMAssay Description:Binding affinity to N-terminal 6His-tagged GDP-bound Galphai1 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetGuanine nucleotide-binding protein G(i) subunit alpha-1(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50617967(CHEMBL5434513)
Affinity DataKd:  2.55E+4nMAssay Description:Binding affinity to N-terminal 6His-tagged GDP-bound Galphai1 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed