Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50020287
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 0.810nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 0.850nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 8.5nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 8.60nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Human)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]CP55490 from CB2 receptor (unknown origin) expressed in CHO-K1 cells by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Human)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]CP55490 from CB2 receptor (unknown origin) expressed in CHO-K1 cells by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 138nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 171nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 193nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism (NIAAA)
Curated by ChEMBL
Affinity DataKi: 203nMAssay Description:Displacement of [3H]CP55490 from CB1 receptor in mouse brain plasma membrane by radioligand displacement analysisMore data for this Ligand-Target Pair















































