Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50020289
TargetKappa-type opioid receptor(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50002184(Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Ly...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]diprenorphine from mouse KOR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50628568(CHEMBL5438249)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]diprenorphine from mouse KOR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50628570(CHEMBL5417671)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]diprenorphine from mouse KOR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50628565(CHEMBL5428690)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]diprenorphine from mouse KOR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50628566(CHEMBL5429387)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]diprenorphine from mouse KOR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50628569(CHEMBL5401977)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]diprenorphine from mouse KOR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Mouse)
Medical University of Vienna

Curated by ChEMBL
LigandPNGBDBM50628567(CHEMBL5407015)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]diprenorphine from mouse KOR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by radioligand ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed