Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50020330
Affinity DataKd: 25nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 34nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 41nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 41nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 45nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 53nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 63nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 66nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 72nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 73nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Binding affinity to VHL/Elongin B/Elongin C (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 86nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 90nMAssay Description:Binding affinity to VHL/Elongin B/Elongin C (unknown origin) using FAM-DEALA-Hyp-YIPMDDDFQLRSF as substrate assessed as dissociation constant by fluo...More data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 112nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in permeabilized HEK293 cells using NanoGlo substrate incubated for 30 mins by tracer ba...More data for this Ligand-Target Pair
Affinity DataIC50: 122nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in permeabilized HEK293 cells using NanoGlo substrate incubated for 30 mins by tracer ba...More data for this Ligand-Target Pair
Affinity DataKd: 129nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 134nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 141nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 149nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 162nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 163nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 164nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo substrate incubated for 30 mins by tracer based NanoB...More data for this Ligand-Target Pair
Affinity DataKd: 183nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 186nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 213nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in permeabilized HEK293 cells using NanoGlo substrate incubated for 30 mins by tracer ba...More data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 244nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B (1 to 104 residues)/Elongin C (17 to 112 residues) (unknown origin) exp...More data for this Ligand-Target Pair
Affinity DataKd: 245nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 268nMAssay Description:Binding affinity to VHL (54 to 213 residues)/N-terminal Avi-tagged biotinylated-Elongin B (1 to 104 residues)/Elongin C (17 to 112 residues) (unknown...More data for this Ligand-Target Pair
Affinity DataKd: 281nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 297nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 305nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo substrate incubated for 30 mins by tracer based NanoB...More data for this Ligand-Target Pair
Affinity DataKd: 322nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 330nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 366nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo substrate incubated for 30 mins by tracer based NanoB...More data for this Ligand-Target Pair
Affinity DataKd: 397nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 496nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 528nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 576nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in permeabilized HEK293 cells using NanoGlo substrate incubated for 30 mins by tracer ba...More data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of NanoLuc-fused VHL (unknown origin) transfected in live HEK293 cells using NanoGlo substrate incubated for 30 mins by tracer based NanoB...More data for this Ligand-Target Pair
Affinity DataKd: 883nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of VHL/Elongin B/Elongin C (unknown origin) using FAM-DEALA-Hyp-YIPD as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.04E+3nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 1.27E+3nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair































