Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50022424
TargetDual specificity protein kinase CLK2(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 122nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 143nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 167nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 173nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 188nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 193nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 194nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 208nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 278nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 296nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 412nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 415nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 445nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 595nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 597nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 685nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 731nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 771nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 790nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 877nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 949nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform epsilon(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CK1epsilon (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+3nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.48E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.97E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.89E+3nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 5.35E+3nMAssay Description:Inhibition of CLK1 (unknown origin)More data for this Ligand-Target Pair






