Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50048711
TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50007407(1-NP | 1-Naphthalen-1-yl-piperazine | 4-Naphthalen...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50007411(1-Naphthalen-2-yl-piperazine | CHEMBL278509)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50025465(8-Methoxy-2-piperazin-1-yl-quinoline | 8-Methoxyqu...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50025469(8-Methoxy-2-(4-methyl-piperazin-1-yl)-quinoline | ...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50001898(1-Phenyl-piperazine | CHEMBL9434 | PHENYLPIPERAZIN...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM23981((2S)-1,2,3,4-Tetrahydro-naphthalen-2-ylamine | 1,2...)
Affinity DataKi:  1.11E+4nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50025466(8-Methoxy-quinolin-2-ylamine | CHEMBL77072)
Affinity DataKi:  3.50E+4nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50025467(2-(N-dipropylamino)quinoline | CHEMBL78878 | Dipro...)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50226052(CHEMBL80988)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50226053(CHEMBL75983)
Affinity DataKi:  7.10E+4nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM14322(2-Aminoquinoline 1 | 2-aminoquinoline | CHEMBL6123...)
Affinity DataKi:  7.90E+4nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50025470(2-Piperidin-1-yl-quinoline | CHEMBL76495 | N4-Deaz...)
Affinity DataKi: >1.50E+5nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetSerotonin 2 (5-HT2) receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50226051(CHEMBL80298 | Quinolin-3-ylamine)
Affinity DataKi: >3.00E+5nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat cortical membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed