Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50019444
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605906BDBM50605906(CHEMBL5172767)
Affinity DataKd:  7.30nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619312BDBM50619312(CHEMBL5399070)
Affinity DataKd:  19nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619313BDBM50619313(CHEMBL5417058)
Affinity DataKd:  48nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619315BDBM50619315(CHEMBL5417476)
Affinity DataKd:  53nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619316BDBM50619316(CHEMBL5439857)
Affinity DataKd:  56nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619314BDBM50619314(CHEMBL5406944)
Affinity DataKd:  62nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50550127BDBM50550127(CHEMBL4781866)
Affinity DataKd:  160nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KdELECT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619317BDBM50619317(CHEMBL5416400)
Affinity DataKd:  165nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50572241BDBM50572241(DNDI1417016 | CHEMBL2094383)
Affinity DataKd:  200nMAssay Description:Binding affinity to human RIOK2 assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605905BDBM50605905(CHEMBL5184068)
Affinity DataKd: <200nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31095BDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd: <200nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 4814BDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd: <200nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619311BDBM50619311(CHEMBL5411549)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50619318BDBM50619318(CHEMBL5424801)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to RIOK2 (unknown origin) assessed as dissociation constant by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase RIO2(Human)
Jinan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50550133BDBM50550133(CHEMBL4754518)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of NLuc-tagged RIOK2 (unknown origin) transfected in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed