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Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50020846
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50591962(CHEMBL5175418)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of PAK4 (unknown origin) using S2 substrate incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM101618(US8530652, 114)
Affinity DataIC50: 9nMAssay Description:Inhibition of PAK4 (unknown origin) using lipid substrate incubated for 40 mins in presence of ATP by ADP-Glo plus luminescence kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50634059(CHEMBL5429021)
Affinity DataIC50: 9nMAssay Description:Inhibition of PAK4 (unknown origin) using lipid substrate incubated for 40 mins in presence of ATP by ADP-Glo plus luminescence kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50634054(CHEMBL5411182)
Affinity DataIC50: 10nMAssay Description:Inhibition of PAK4 (unknown origin) using lipid substrate incubated for 40 mins in presence of ATP by ADP-Glo plus luminescence kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50634058(CHEMBL5400697)
Affinity DataIC50: 11nMAssay Description:Inhibition of PAK4 (unknown origin) using lipid substrate incubated for 40 mins in presence of ATP by ADP-Glo plus luminescence kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50634056(CHEMBL5395115)
Affinity DataIC50: 13nMAssay Description:Inhibition of PAK4 (unknown origin) using lipid substrate incubated for 40 mins in presence of ATP by ADP-Glo plus luminescence kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50634055(CHEMBL5414332)
Affinity DataIC50: 16nMAssay Description:Inhibition of PAK4 (unknown origin) using lipid substrate incubated for 40 mins in presence of ATP by ADP-Glo plus luminescence kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM101618(US8530652, 114)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant human N-terminal 6His-tagged PAK4 kinase domain (300 to 591 residues) incubated in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50634057(CHEMBL5401120)
Affinity DataIC50: 24nMAssay Description:Inhibition of PAK4 (unknown origin) using lipid substrate incubated for 40 mins in presence of ATP by ADP-Glo plus luminescence kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50634060(CHEMBL5438274)
Affinity DataIC50: 100nMAssay Description:Inhibition of PAK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed