Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50020863
TargetGTPase KRas(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50634302(CHEMBL5417773)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human GTP-bound KRAS wild type (1 to 169 residues) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetGTPase KRas(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50634304(CHEMBL5398447)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human GTP-bound KRAS wild type (1 to 169 residues) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetGTPase KRas(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50585402(CHEMBL5081048)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human GTP-bound KRAS wild type (1 to 169 residues) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetGTPase KRas(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50634305(CHEMBL5434863)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant human GTP-bound KRAS wild type (1 to 169 residues) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetGTPase KRas(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50634303(CHEMBL5429156)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human GTP-bound KRAS wild type (1 to 169 residues) incubated for 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed