Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50021502
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641339(CHEMBL5567027)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50605682(CHEMBL5176915)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641324(CHEMBL5595401)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641327(CHEMBL5567389)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641340(CHEMBL5570158)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641323(CHEMBL5590627)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641326(CHEMBL5571621)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641329(CHEMBL5574704)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641332(CHEMBL5549926)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641328(CHEMBL5573282)
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641333(CHEMBL5575182)
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641325(CHEMBL5549920)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641334(CHEMBL5563136)
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM60622(BDBM50300355 | US9133148, A | US11753371, Compound...)
Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641330(CHEMBL5593092)
Affinity DataIC50: 49nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641331(CHEMBL5570616)
Affinity DataIC50: 61nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641336(CHEMBL5565395)
Affinity DataIC50: 112nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641337(CHEMBL5574429)
Affinity DataIC50: 149nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641327(CHEMBL5567389)
Affinity DataIC50: 193nMAssay Description:Reversible inhibition of MAGL in human U-937 cells using 2-oleoylglycerol as substrate preincubated with compound for 30 mins followed by substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641324(CHEMBL5595401)
Affinity DataIC50: 197nMAssay Description:Reversible inhibition of MAGL in human U-937 cells using 2-oleoylglycerol as substrate preincubated with compound for 30 mins followed by substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641339(CHEMBL5567027)
Affinity DataIC50: 199nMAssay Description:Reversible inhibition of MAGL in human U-937 cells using 2-oleoylglycerol as substrate preincubated with compound for 30 mins followed by substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641335(CHEMBL5564512)
Affinity DataIC50: 242nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641340(CHEMBL5570158)
Affinity DataIC50: 489nMAssay Description:Reversible inhibition of MAGL in human U-937 cells using 2-oleoylglycerol as substrate preincubated with compound for 30 mins followed by substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50641338(CHEMBL5570539)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant MAGL using 4-nitrophenylacetate as substrate incubated for 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed