Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50021926
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding affinity to STAT3 SH2 domain (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 (127 to 711 residues) DNA-binding activity transfected...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C468A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C542S mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C468A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 (127 to 711 residues) DNA-binding activity transfected...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 (127 to 711 residues) DNA-binding activity transfected...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C328A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 (127 to 711 residues) DNA-binding activity transfected...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C542S mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C426A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C328A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C542S mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C542S mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C426A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C328A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 8.60E+3nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C328A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 9.70E+3nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C426A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C328A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 (127 to 711 residues) DNA-binding activity transfected...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.45E+4nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) DNA-binding activity transfected in v-Src transformed mouse NIH3T3...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.89E+4nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C426A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.01E+4nMAssay Description:Inhibition of recombinant wild type tyrosine phosphorylated C-terminal 6His tagged human STAT3 C468A mutant (127 to 711 residues) DNA-binding activit...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.01E+4nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.03E+4nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Human)
Cedars-Sinai Medical Center
Curated by ChEMBL
Cedars-Sinai Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.16E+4nMAssay Description:Displacement of 5-carboxyfluorescein GpYLPQTV-NH2 probe from C-terminal 6His-tagged recombinant human STAT3 (127 to 711 residues) SH2 domain extracte...More data for this Ligand-Target Pair







