Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50020556
TargetMu-type opioid receptor(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631210BDBM50631210(CHEMBL5415173)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor (unknown origin) expressed in CHO cell membrane measured after 90 mins by beta-scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590799BDBM50590799(CHEMBL5179132)
Affinity DataKi:  36nMAssay Description:Antagonist activity at sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514276BDBM50514276(CHEMBL4439908)
Affinity DataKi:  57nMAssay Description:Antagonist activity at sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514245BDBM50514245(CHEMBL4461774)
Affinity DataKi:  58nMAssay Description:Antagonist activity at sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608017BDBM50608017(CHEMBL5287561)
Affinity DataKi: <100nMAssay Description:Antagonist activity at sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580843BDBM50580843(CHEMBL5086571)
Affinity DataKi:  108nMAssay Description:Antagonist activity at sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548568BDBM50548568(CHEMBL4781352)
Affinity DataKi:  118nMAssay Description:Antagonist activity at sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590776BDBM50590776(CHEMBL172155)
Affinity DataKi:  241nMAssay Description:Antagonist activity at sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631210BDBM50631210(CHEMBL5415173)
Affinity DataKi:  364nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631210BDBM50631210(CHEMBL5415173)
Affinity DataKi:  877nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane in presence of sigma1 receptor agonist, phenytoin by radioligand b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
Sichuan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631211BDBM50631211(CHEMBL5418375)
Affinity DataKi:  8.30E+3nMAssay Description:Displacement of [3H]-pentazocine from sigma1 receptor in guinea pig brain membrane by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed