Compile Data Set for Download or QSAR
Report error Found 81 Enz. Inhib. hit(s) with all data for entry = 50021522
LigandPNGBDBM50598851(CHEMBL5199076 | US20240207300, Compound 292)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743588(US20250163077, Example 14)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743604(US20250163077, Example 30)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50598844(CHEMBL5200005 | US12435090, Compound 164)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743587(US20250163077, Example 13)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743578(US20250163077, Example 4)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743577(US20250163077, Example 3)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641505(CHEMBL5573390)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641504(CHEMBL5567277)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743594(US20250163077, Example 20)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743606(US20250163077, Example 32)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743597(US20250163077, Example 23)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743596(US20250163077, Example 22)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743575(US20250163077, Example 1)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743591(US20250163077, Example 17)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743611(US20250163077, Example 37)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743609(US20250163077, Example 35)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743595(US20250163077, Example 21)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743598(US20250163077, Example 24)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641510(CHEMBL5566287)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743599(US20250163077, Example 25)
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM3096(6-(2,6-dichlorophenyl)-2-({4-[2-(diethylamino)etho...)
Affinity DataIC50: 24nMAssay Description:Inhibition of MYT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641508(CHEMBL5571632)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743582(US20250163077, Example 8)
Affinity DataIC50: 49nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50598851(CHEMBL5199076 | US20240207300, Compound 292)
Affinity DataIC50: 52nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743588(US20250163077, Example 14)
Affinity DataIC50: 63nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743608(US20250163077, Example 34)
Affinity DataIC50: 69nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetWee1-like protein kinase(Human)TBA
LigandPNGBDBM3096(6-(2,6-dichlorophenyl)-2-({4-[2-(diethylamino)etho...)
Affinity DataIC50: 72nMAssay Description:Inhibition of Wee1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM743605(US20250163077, Example 31)
Affinity DataIC50: 92nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetWee1-like protein kinase(Human)TBA
LigandPNGBDBM50192349(9-HYDROXY-4-PHENYLPYRROLO[3,4-C]CARBAZOLE-1,3(2H,6...)
Affinity DataIC50: 97nMAssay Description:Inhibition of Wee1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetWee1-like protein kinase(Human)TBA
LigandPNGBDBM50598851(CHEMBL5199076 | US20240207300, Compound 292)
Affinity DataIC50: 104nMAssay Description:Inhibition of human recombinant Wee1 preincubated with compound for for 15 mins followed by ATP addition and measured after 60 mins by ADP Glo lumine...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetWee1-like protein kinase(Human)TBA
LigandPNGBDBM50598844(CHEMBL5200005 | US12435090, Compound 164)
Affinity DataIC50: 152nMAssay Description:Inhibition of human recombinant Wee1 preincubated with compound for for 15 mins followed by ATP addition and measured after 60 mins by ADP Glo lumine...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743613(US20250163077, Example 39)
Affinity DataIC50: 223nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM31089(DASATINIB)
Affinity DataIC50: 226nMAssay Description:Inhibition of MYT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743587(US20250163077, Example 13)
Affinity DataIC50: 268nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743606(US20250163077, Example 32)
Affinity DataIC50: 271nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641504(CHEMBL5567277)
Affinity DataIC50: 289nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641505(CHEMBL5573390)
Affinity DataIC50: 293nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743597(US20250163077, Example 23)
Affinity DataIC50: 334nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743591(US20250163077, Example 17)
Affinity DataIC50: 358nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743610(US20250163077, Example 36)
Affinity DataIC50: 359nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743578(US20250163077, Example 4)
Affinity DataIC50: 420nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743594(US20250163077, Example 20)
Affinity DataIC50: 578nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743596(US20250163077, Example 22)
Affinity DataIC50: 660nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743595(US20250163077, Example 21)
Affinity DataIC50: 705nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641507(CHEMBL5570533)
Affinity DataIC50: 714nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641506(CHEMBL5572096)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641509(CHEMBL5593294)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human recombinant MYT1 incubated for 60 mins in presence of tracer178 by HTRF analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50641508(CHEMBL5571632)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM743609(US20250163077, Example 35)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of CDK1 phosphorylation at Thr14 residue in human HCC1569 cells incubated for 6 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
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