Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50021757
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of 15-LOX (unknown origin)More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of 15-LOX (unknown origin)More data for this Ligand-Target Pair
TargetCystine/glutamate transporter(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of Xc- in human HT-1080 cells assessed as decrease in glutamate release incubated for 2 hrs by Amplex red assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of 15-LOX (unknown origin)More data for this Ligand-Target Pair
TargetAcetyl-CoA acetyltransferase, cytosolic(Homo sapiens)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of Acetyl-CoA acetyltransferase (unknown origin)More data for this Ligand-Target Pair
TargetAcetyl-CoA acetyltransferase, cytosolic(Homo sapiens)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of Acetyl-CoA acetyltransferase (unknown origin)More data for this Ligand-Target Pair
TargetAcetyl-CoA acetyltransferase, cytosolic(Homo sapiens)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Acetyl-CoA acetyltransferase (unknown origin)More data for this Ligand-Target Pair
TargetCystine/glutamate transporter(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Xc- in human HT-1080 cells assessed as decrease in glutamate release incubated for 2 hrs by Amplex red assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of 15-LOX (unknown origin)More data for this Ligand-Target Pair
TargetCystine/glutamate transporter(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Xc- in human HT-1080 cells assessed as decrease in glutamate release incubated for 2 hrs by Amplex red assayMore data for this Ligand-Target Pair
TargetAcetyl-CoA acetyltransferase, cytosolic(Homo sapiens)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 171nMAssay Description:Inhibition of Acetyl-CoA acetyltransferase (unknown origin)More data for this Ligand-Target Pair
TargetAcetyl-CoA acetyltransferase, cytosolic(Homo sapiens)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 269nMAssay Description:Inhibition of Acetyl-CoA acetyltransferase (unknown origin)More data for this Ligand-Target Pair
TargetCystine/glutamate transporter(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of Xc- in human HT-1080 cells assessed as decrease in glutamate release incubated for 2 hrs by Amplex red assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of 15-LOX (unknown origin)More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 950nMAssay Description:Inhibition of 15-LOX (unknown origin)More data for this Ligand-Target Pair
TargetAcetyl-CoA acetyltransferase, cytosolic(Homo sapiens)
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Indian Institute of Technology (Banaras Hindu University)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Acetyl-CoA acetyltransferase (unknown origin)More data for this Ligand-Target Pair















