Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50021618
TargetProbable global transcription activator SNF2L2(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642737(CHEMBL5564941)
Affinity DataIC50: 1.20nMAssay Description:Binding affinity to his-tagged BRM bromodomain (unknown origin) by alpha-LISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642738(CHEMBL5571722)
Affinity DataIC50: 2.70nMAssay Description:Binding affinity to his-tagged BRM bromodomain (unknown origin) by alpha-LISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642738(CHEMBL5571722)
Affinity DataIC50: 2.80nMAssay Description:Binding affinity to his-tagged BRG1 bromodomain (unknown origin) by alpha-LISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642737(CHEMBL5564941)
Affinity DataIC50: 3.30nMAssay Description:Binding affinity to his-tagged BRG1 bromodomain (unknown origin) by alpha-LISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642739(CHEMBL5575147)
Affinity DataKd:  3.40nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642736(CHEMBL5574201)
Affinity DataIC50: 16nMAssay Description:Binding affinity to his-tagged BRG1 bromodomain (unknown origin) by alpha-LISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642736(CHEMBL5574201)
Affinity DataIC50: 18nMAssay Description:Binding affinity to his-tagged BRM bromodomain (unknown origin) by alpha-LISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642740(CHEMBL5565613)
Affinity DataKd:  65nMAssay Description:Binding affinity to his-tagged BRG1 bromodomain (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642739(CHEMBL5575147)
Affinity DataKd:  72nMAssay Description:Binding affinity to his-tagged BRM bromodomain (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642740(CHEMBL5565613)
Affinity DataKd:  93nMAssay Description:Binding affinity to his-tagged BRM bromodomain (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642739(CHEMBL5575147)
Affinity DataKd:  108nMAssay Description:Binding affinity to his-tagged BRG1 bromodomain (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642740(CHEMBL5565613)
Affinity DataKd:  350nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642744(CHEMBL5566479)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
Targetvon Hippel-Lindau disease tumor suppressor(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642743(CHEMBL5595617)
Affinity DataKd:  4.70E+3nMAssay Description:Binding affinity to VHL (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642742(CHEMBL5569524)
Affinity DataKd:  5.22E+3nMAssay Description:Binding affinity to his-tagged BRG1 bromodomain (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642742(CHEMBL5569524)
Affinity DataKd:  8.54E+3nMAssay Description:Binding affinity to his-tagged BRM bromodomain (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProbable global transcription activator SNF2L2(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642741(CHEMBL5573721)
Affinity DataKd:  1.03E+4nMAssay Description:Binding affinity to his-tagged BRM bromodomain (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTranscription activator BRG1(Human)
Arvinas LLC

Curated by ChEMBL
LigandPNGBDBM50642741(CHEMBL5573721)
Affinity DataKd:  1.26E+4nMAssay Description:Binding affinity to his-tagged BRG1 bromodomain (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed