Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50021631
TargetNeutral amino acid transporter B(0)(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50642838(CHEMBL5570488)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of ASCT2 in HEK293 cells assessed as reduction in glutamine uptake preincubated for 5 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNeutral amino acid transporter B(0)(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50642839(CHEMBL5572948)
Affinity DataIC50: 5.14E+3nMAssay Description:Inhibition of ASCT2 in HEK293 cells assessed as reduction in glutamine uptake preincubated for 5 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNeutral amino acid transporter B(0)(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50642837(CHEMBL5569240)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of ASCT2 in HEK293 cells assessed as reduction in glutamine uptake preincubated for 5 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNeutral amino acid transporter B(0)(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50642838(CHEMBL5570488)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of ASCT2 in human A549 cells assessed as reduction in glutamine uptake preincubated for 5 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNeutral amino acid transporter B(0)(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50642839(CHEMBL5572948)
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibition of ASCT2 in human A549 cells assessed as reduction in glutamine uptake preincubated for 5 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNeutral amino acid transporter B(0)(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50140122(CHEMBL3754053)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of ASCT2 in HEK293 cells assessed as reduction in glutamine uptake preincubated for 5 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed