Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50022014
TargetMu-type opioid receptor(Human)TBA
LigandPNGBDBM50647255(CHEMBL5589843)
Affinity DataKi:  0.820nMAssay Description:Displacement of [3H]-DAMGO from human MOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647255(CHEMBL5589843)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]U-69593 from human KOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647257(CHEMBL5596704)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]U-69593 from human KOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647255(CHEMBL5589843)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]DPDPE from human DOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMu-type opioid receptor(Human)TBA
LigandPNGBDBM50647256(CHEMBL5597092)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-DAMGO from human MOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647256(CHEMBL5597092)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]U-69593 from human KOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMu-type opioid receptor(Human)TBA
LigandPNGBDBM50647257(CHEMBL5596704)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-DAMGO from human MOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647257(CHEMBL5596704)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPDPE from human DOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMu-type opioid receptor(Human)TBA
LigandPNGBDBM50647261(CHEMBL5596729)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]-DAMGO from human MOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647256(CHEMBL5597092)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]DPDPE from human DOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMu-type opioid receptor(Human)TBA
LigandPNGBDBM50647262(CHEMBL5598475)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]-DAMGO from human MOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647261(CHEMBL5596729)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]U-69593 from human KOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMu-type opioid receptor(Human)TBA
LigandPNGBDBM50647258(CHEMBL5596196)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-DAMGO from human MOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647258(CHEMBL5596196)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]DPDPE from human DOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647260(CHEMBL5590334)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]U-69593 from human KOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647258(CHEMBL5596196)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]U-69593 from human KOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647261(CHEMBL5596729)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]DPDPE from human DOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMu-type opioid receptor(Human)TBA
LigandPNGBDBM50647260(CHEMBL5590334)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]-DAMGO from human MOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647262(CHEMBL5598475)
Affinity DataKi:  390nMAssay Description:Displacement of [3H]U-69593 from human KOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647262(CHEMBL5598475)
Affinity DataKi:  620nMAssay Description:Displacement of [3H]DPDPE from human DOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMu-type opioid receptor(Human)TBA
LigandPNGBDBM50647259(CHEMBL5590096)
Affinity DataKi:  690nMAssay Description:Displacement of [3H]-DAMGO from human MOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647259(CHEMBL5590096)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]DPDPE from human DOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647259(CHEMBL5590096)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]U-69593 from human KOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50647260(CHEMBL5590334)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from human DOR extracted from HEK293 cell membrane assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed