Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50020070
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataKi:  40nMAssay Description:Binding affinity to electric eel AChE assessed as inhibition constant by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 50nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625941(CHEMBL5435446)
Affinity DataIC50: 60nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625931(CHEMBL5411326)
Affinity DataIC50: 120nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625931(CHEMBL5411326)
Affinity DataKi:  170nMAssay Description:Binding affinity to electric eel AChE assessed as inhibition constant by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625940(CHEMBL5397094)
Affinity DataIC50: 180nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625941(CHEMBL5435446)
Affinity DataKi:  220nMAssay Description:Binding affinity to electric eel AChE assessed as inhibition constant by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625936(CHEMBL5401023)
Affinity DataKi:  270nMAssay Description:Binding affinity to electric eel AChE assessed as inhibition constant by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625944(CHEMBL5415333)
Affinity DataIC50: 280nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625930(CHEMBL5420759)
Affinity DataIC50: 350nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625936(CHEMBL5401023)
Affinity DataIC50: 370nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625933(CHEMBL5413249)
Affinity DataIC50: 410nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625945(CHEMBL5423996)
Affinity DataIC50: 440nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625934(CHEMBL5433803)
Affinity DataIC50: 450nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625935(CHEMBL5418957)
Affinity DataIC50: 660nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625940(CHEMBL5397094)
Affinity DataIC50: 710nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625938(CHEMBL5421487)
Affinity DataIC50: 750nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625939(CHEMBL5405227)
Affinity DataIC50: 800nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625943(CHEMBL5396980)
Affinity DataIC50: 960nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625939(CHEMBL5405227)
Affinity DataIC50: 970nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625930(CHEMBL5420759)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625934(CHEMBL5433803)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625933(CHEMBL5413249)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625938(CHEMBL5421487)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625945(CHEMBL5423996)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625942(CHEMBL5397579)
Affinity DataKi:  1.65E+3nMAssay Description:Binding affinity to electric eel AChE assessed as inhibition constant by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625941(CHEMBL5435446)
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625943(CHEMBL5396980)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625942(CHEMBL5397579)
Affinity DataIC50: 2.49E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625932(CHEMBL5401594)
Affinity DataKi:  2.57E+3nMAssay Description:Binding affinity to electric eel AChE assessed as inhibition constant by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625944(CHEMBL5415333)
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625942(CHEMBL5397579)
Affinity DataIC50: 2.94E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625935(CHEMBL5418957)
Affinity DataIC50: 4.73E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625931(CHEMBL5411326)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625932(CHEMBL5401594)
Affinity DataIC50: 4.95E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625937(CHEMBL5435159)
Affinity DataKi:  6.87E+3nMAssay Description:Binding affinity to electric eel AChE assessed as inhibition constant by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625932(CHEMBL5401594)
Affinity DataIC50: 7.15E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625936(CHEMBL5401023)
Affinity DataIC50: 8.58E+3nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625937(CHEMBL5435159)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM50625937(CHEMBL5435159)
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetCholinesterase(Horse)
Chulabhorn Research Institute

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of horse serum BuChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed