Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50021689
TargetCathepsin D(Human)TBA
LigandPNGBDBM50643516(CHEMBL5569371)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human Cathepsin D using MCA labeled GKPILFFRLK(DNP)-D-R-NH2 as substrate preincubated for 10 mins followed by substrate addition by FRE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCathepsin D(Human)TBA
LigandPNGBDBM50643518(CHEMBL5571122)
Affinity DataIC50: 2nMAssay Description:Inhibition of human Cathepsin D using MCA labeled GKPILFFRLK(DNP)-D-R-NH2 as substrate preincubated for 10 mins followed by substrate addition by FRE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCathepsin D(Human)TBA
LigandPNGBDBM50025902(3-Hydroxy-4-[2-(3-hydroxy-6-methyl-4-{3-methyl-2-[...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human Cathepsin D using MCA labeled GKPILFFRLK(DNP)-D-R-NH2 as substrate preincubated for 10 mins followed by substrate addition by FRE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCathepsin D(Human)TBA
LigandPNGBDBM50643514(CHEMBL5570548)
Affinity DataIC50: 28nMAssay Description:Inhibition of human Cathepsin D using MCA labeled GKPILFFRLK(DNP)-D-R-NH2 as substrate preincubated for 10 mins followed by substrate addition by FRE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCathepsin D(Human)TBA
LigandPNGBDBM50643515(CHEMBL5573834)
Affinity DataIC50: 58nMAssay Description:Inhibition of human Cathepsin D using MCA labeled GKPILFFRLK(DNP)-D-R-NH2 as substrate preincubated for 10 mins followed by substrate addition by FRE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCathepsin D(Human)TBA
LigandPNGBDBM50643513(CHEMBL5594826)
Affinity DataIC50: 65nMAssay Description:Inhibition of human Cathepsin D using MCA labeled GKPILFFRLK(DNP)-D-R-NH2 as substrate preincubated for 10 mins followed by substrate addition by FRE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCathepsin D(Human)TBA
LigandPNGBDBM50643517(CHEMBL5569502)
Affinity DataIC50: 72nMAssay Description:Inhibition of human Cathepsin D using MCA labeled GKPILFFRLK(DNP)-D-R-NH2 as substrate preincubated for 10 mins followed by substrate addition by FRE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCathepsin D(Human)TBA
LigandPNGBDBM50643512(CHEMBL5572049)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human Cathepsin D using MCA labeled GKPILFFRLK(DNP)-D-R-NH2 as substrate preincubated for 10 mins followed by substrate addition by FRE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed