Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50021690
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643552(CHEMBL5572902)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50462572(CHEMBL4249337)
Affinity DataIC50: 9nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643520(CHEMBL5570019)
Affinity DataIC50: 13nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643550(CHEMBL5564160)
Affinity DataIC50: 17nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643523(CHEMBL5595468)
Affinity DataIC50: 18nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643522(CHEMBL5570786)
Affinity DataIC50: 29nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643546(CHEMBL5589648)
Affinity DataIC50: 41nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643551(CHEMBL5570295)
Affinity DataIC50: 81nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643553(CHEMBL5594911)
Affinity DataIC50: 86nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643526(CHEMBL5575577)
Affinity DataIC50: 89nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643532(CHEMBL5564069)
Affinity DataIC50: 89nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643543(CHEMBL5579716)
Affinity DataIC50: 91nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643544(CHEMBL5593189)
Affinity DataIC50: 126nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643528(CHEMBL5590530)
Affinity DataIC50: 226nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643534(CHEMBL5574155)
Affinity DataIC50: 226nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643524(CHEMBL5591696)
Affinity DataIC50: 234nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643547(CHEMBL5593229)
Affinity DataIC50: 279nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643548(CHEMBL5562894)
Affinity DataIC50: 340nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643542(CHEMBL5569153)
Affinity DataIC50: 344nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643527(CHEMBL5574353)
Affinity DataIC50: 358nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643533(CHEMBL5567163)
Affinity DataIC50: 358nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643545(CHEMBL5573050)
Affinity DataIC50: 365nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643549(CHEMBL5563082)
Affinity DataIC50: 379nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643541(CHEMBL5571402)
Affinity DataIC50: 456nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643519(CHEMBL5563557)
Affinity DataIC50: 497nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643521(CHEMBL5566597)
Affinity DataIC50: 721nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643540(CHEMBL5568753)
Affinity DataIC50: 918nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643525(CHEMBL5565586)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643530(CHEMBL5564112)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643529(CHEMBL5570599)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643531(CHEMBL5574244)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643537(CHEMBL5595149)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643536(CHEMBL5565719)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643535(CHEMBL5575956)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643520(CHEMBL5570019)
Affinity DataIC50: 2.82E+3nMAssay Description:Inhibition of PRMT1 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643539(CHEMBL5568905)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643538(CHEMBL5590990)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PRMT5 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643520(CHEMBL5570019)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of PRMT4 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643526(CHEMBL5575577)
Affinity DataIC50: 6.89E+3nMAssay Description:Inhibition of PRMT1 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643520(CHEMBL5570019)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PRMT8 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643526(CHEMBL5575577)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PRMT4 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase NSD3(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643520(CHEMBL5570019)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of NSD3 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643526(CHEMBL5575577)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of NSD2 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643520(CHEMBL5570019)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of NSD2 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643526(CHEMBL5575577)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PRMT8 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643526(CHEMBL5575577)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of EZH2 (unknown origin) using SAM and peptide substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643520(CHEMBL5570019)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of EZH2 (unknown origin) using SAM and peptide substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase NSD3(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50643526(CHEMBL5575577)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of NSD3 methyltransferase activity (unknown origin) using histone H4/SAM as substrate incubated for 80 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed