Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50021657
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643185(CHEMBL5572737 | US20250243196, Compound F-90)
Affinity DataKd:  0.300nMAssay Description:Binding affinity to NanoLuc fused-CITK kinase domain (unknown origin) expressed in HEK293T cells assessed as dissociation constant NanoBRET Target En...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643187(CHEMBL5591534 | US20250243196, Compound F-162)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643185(CHEMBL5572737 | US20250243196, Compound F-90)
Affinity DataKd:  9.5nMAssay Description:Binding affinity to NanoLuc fused-CITK (unknown origin) expressed in HEK293T cells assessed as dissociation constant NanoBRET Target Engagement Intra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643156(CHEMBL5568742 | US20250243196, Compound F-21)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643185(CHEMBL5572737 | US20250243196, Compound F-90)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643144(CHEMBL5595104 | US20250243196, Compound F-9)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643157(CHEMBL5575901 | US20250243196, Compound F-16)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643161(CHEMBL5569359 | US20250243196, Compound F-58)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643136(CHEMBL5579704 | US20250243196, Compound F-13)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643188(CHEMBL5575300 | US20250243196, Compound F-161)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643183(CHEMBL5595678 | US20250243196, Compound F-57)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643164(CHEMBL5590268 | US20250243196, Compound F-62)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643184(CHEMBL5575657 | US20250243196, Compound F-89)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643180(CHEMBL5574799 | US20250243196, Compound F-48)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643146(CHEMBL5566667 | US20250243196, Compound F-41)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643153(CHEMBL5562828 | US20250243196, Compound F-17)
Affinity DataIC50: 31nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643166(CHEMBL5566783 | US20250243196, Compound F-80)
Affinity DataIC50: 31nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643169(CHEMBL5574511 | US20250243196, Compound F-81)
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643163(CHEMBL5542511 | US20250243196, Compound F-65)
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643178(CHEMBL5573191)
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643171(CHEMBL5563128 | US20250243196, Compound F-83)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643138(CHEMBL5571250 | US20250243196, Compound F-33)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643158(CHEMBL5574143 | US20250243196, Compound F-77)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643142(CHEMBL5571047 | US20250243196, Compound F-40)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643145(CHEMBL5572919 | US20250243196, Compound F-8)
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643181(CHEMBL5563995 | US20250243196, Compound F-53)
Affinity DataIC50: 48nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643182(CHEMBL5574850 | US20250243196, Compound F-55)
Affinity DataIC50: 54nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643155(CHEMBL5570381 | US20250243196, Compound F-20)
Affinity DataIC50: 61nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643135(CHEMBL5590500 | US20250243196, Compound F-7)
Affinity DataIC50: 66nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643179(CHEMBL5574584 | US20250243196, Compound F-106)
Affinity DataIC50: 67nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643160(CHEMBL5566515 | US20250243196, Compound F-75)
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643162(CHEMBL5566014 | US20250243196, Compound F-78)
Affinity DataIC50: 89nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643143(CHEMBL5571741 | US20250243196, Compound F-36)
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643175(CHEMBL5572680 | US20250243196, Compound F-110)
Affinity DataIC50: 92nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643168(CHEMBL5590585 | US20250243196, Compound F-67)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643174(CHEMBL5575031 | US20250243196, Compound F-85)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643159(CHEMBL5583840 | US20250243196, Compound F-61)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50319005((R)-4-(1-aminoethyl)-N-(1H-pyrrolo[2,3-b]pyridin-4...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643173(CHEMBL5575191 | US20250243196, Compound F-84)
Affinity DataIC50: 160nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643154(CHEMBL5564045 | US20250243196, Compound F-19)
Affinity DataIC50: 160nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643170(CHEMBL5566310 | US20250243196, Compound F-68)
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643167(CHEMBL5569087 | US20250243196, Compound F-79)
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAP2-associated protein kinase 1(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643185(CHEMBL5572737 | US20250243196, Compound F-90)
Affinity DataIC50: 212nMAssay Description:Inhibition of human AAK1 incubated for 120 mins by [33P]-gammaATP based Radiometric scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643130(CHEMBL5574968)
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643147(CHEMBL5571124 | US20250243196, Compound F-42)
Affinity DataIC50: 280nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643137(CHEMBL5595129 | US20250243196, Compound F-11)
Affinity DataIC50: 320nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643140(CHEMBL5574306 | US20250243196, Compound F-38)
Affinity DataIC50: 330nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643172(CHEMBL5565388 | US20250243196, Compound F-86)
Affinity DataIC50: 340nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643151(CHEMBL5574767)
Affinity DataIC50: 410nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCitron Rho-interacting kinase(Human)
Lerner Research Institute

Curated by ChEMBL
LigandPNGBDBM50643129(CHEMBL5571901)
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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