Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50021028
TargetAurora kinase B(Human)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM142744(US8937095, 6)
Affinity DataIC50: 3nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase B(Human)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50636122(CHEMBL5549914)
Affinity DataIC50: 11nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase B(Human)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50636123(CHEMBL5567353)
Affinity DataKi:  20nMAssay Description:Binding affinity to Aurora B (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase B(Human)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM4811((Z)-3-[2,4-dimethyl-5-(2-oxo-1,2-dihydro-indol-3-y...)
Affinity DataIC50: 47nMAssay Description:Inhibition of Aurora B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase A(Human)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM14210(N-[4-({6-methoxy-7-[3-(morpholin-4-yl)propoxy]quin...)
Affinity DataIC50: 110nMAssay Description:Inhibition of N terminal his tagged recombinant Aurora A (unknown origin) expressed in baculovirus expression system incubated for 60 mins in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase B(Human)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM14210(N-[4-({6-methoxy-7-[3-(morpholin-4-yl)propoxy]quin...)
Affinity DataIC50: 130nMAssay Description:Inhibition of N terminal his tagged recombinant Aurora B (unknown origin) expressed in baculovirus expression system incubated for 60 mins in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase B(Human)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50273571(Hesperadin | TCMDC-135395 | N-(2-oxo-3-(phenyl(4-(...)
Affinity DataIC50: 250nMAssay Description:Inhibition of Aurora B in human HeLa cells using histone H1 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase B(Human)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  380nMAssay Description:Binding affinity to Aurora B (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed