Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50021281
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639035(CHEMBL5561508)
Affinity DataEC50:  80nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639035(CHEMBL5561508)
Affinity DataEC50:  90nMAssay Description:Agonist activity at Strongyloides stercoralis DAF-12 LBD transfected in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639036(CHEMBL5558148)
Affinity DataEC50:  410nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639036(CHEMBL5558148)
Affinity DataEC50:  470nMAssay Description:Agonist activity at Strongyloides stercoralis DAF-12 LBD transfected in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639037(CHEMBL5565920)
Affinity DataEC50:  650nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639041(CHEMBL5563296)
Affinity DataEC50:  1.02E+3nMAssay Description:Partial agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639040(CHEMBL5563343)
Affinity DataEC50:  1.02E+3nMAssay Description:Partial agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639038(CHEMBL5557658)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639030(CHEMBL5561671)
Affinity DataIC50: 6.90E+3nMAssay Description:Antagonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639039(CHEMBL5556017)
Affinity DataEC50:  7.20E+3nMAssay Description:Partial agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639031(CHEMBL5556518)
Affinity DataIC50: 7.80E+3nMAssay Description:Antagonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639033(CHEMBL5555626)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639029(CHEMBL5560291)
Affinity DataIC50: 1.68E+4nMAssay Description:Antagonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639034(CHEMBL5567262)
Affinity DataIC50: 1.79E+4nMAssay Description:Antagonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639032(CHEMBL5559892)
Affinity DataIC50: 6.00E+4nMAssay Description:Antagonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639030(CHEMBL5561671)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639029(CHEMBL5560291)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639034(CHEMBL5567262)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639033(CHEMBL5555626)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639032(CHEMBL5559892)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetNuclear hormone receptor isoform A(Strongyloides stercoralis)TBA
LigandPNGBDBM50639031(CHEMBL5556518)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at GST-tagged Strongyloides stercoralis DAF-12 LBD incubated for 0.5 hrs in presence of biotinylated SRC1 and SRC2 by Alphascreen as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed