Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50021167
TargetPyruvate kinase PKLR(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50215545(CHEMBL6338)
Affinity DataIC50: 28nMAssay Description:Inhibition of full length N-terminal His-tagged human PKL (2 to 543 residues) expressed in Escherichia coli by kinase Glo luminescence based plate re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPyruvate kinase PKLR(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM4078(Elagic Acid | CHEMBL6246 | 6,7,13,14-tetrahydroxy-...)
Affinity DataIC50: 32nMAssay Description:Inhibition of full length N-terminal His-tagged human PKL (2 to 543 residues) expressed in Escherichia coli by kinase Glo luminescence based plate re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPyruvate kinase PKLR(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50637646(CHEMBL5556210)
Affinity DataIC50: 70nMAssay Description:Inhibition of full length N-terminal His-tagged human PKL (2 to 543 residues) expressed in Escherichia coli by kinase Glo luminescence based plate re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetInterferon-induced, double-stranded RNA-activated protein kinase(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50637646(CHEMBL5556210)
Affinity DataIC50: 180nMAssay Description:Inhibition of PKR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPyruvate kinase PKLR(Human)
University of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50637647(CHEMBL4754666)
Affinity DataIC50: 410nMAssay Description:Inhibition of full length N-terminal His-tagged human PKL (2 to 543 residues) expressed in Escherichia coli by kinase Glo luminescence based plate re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed