Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50021730
Affinity DataIC50: 0.5nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) by phosphosen-csox ...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) by phosphosen-csox ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) by phosphosen-csox ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human wild type S6K2 using RBER-CHKtide as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity to N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) assessed as i...More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) assessed as i...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human wild type S6K2 using RBER-CHKtide as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Inhibition of full length nanoluc-fused FGFR4 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inhibition of full length nanoluc-fused FGFR4 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant FGFR4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity to N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) assessed as i...More data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:Inhibition of full length nanoluc-fused FGFR4 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 2(Human)
Eberhard Karls University Tubingen
Curated by ChEMBL
Eberhard Karls University Tubingen
Curated by ChEMBL
Affinity DataIC50: 156nMAssay Description:Inhibition of MK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 490nMAssay Description:Inhibition of human FGFR2 in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataEC50: 684nMAssay Description:Inhibition of full length nanoluc-fused FGFR1 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataEC50: 867nMAssay Description:Inhibition of full length nanoluc-fused FGFR1 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataEC50: 867nMAssay Description:Inhibition of full length nanoluc-fused FGFR2 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataEC50: 1.29E+3nMAssay Description:Inhibition of full length nanoluc-fused FGFR2 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataEC50: 1.43E+3nMAssay Description:Inhibition of full length nanoluc-fused FGFR3 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataEC50: 1.78E+3nMAssay Description:Inhibition of full length nanoluc-fused FGFR3 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataEC50: 2.24E+3nMAssay Description:Inhibition of full length nanoluc-fused FGFR3 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataEC50: 2.26E+3nMAssay Description:Inhibition of full length nanoluc-fused FGFR4 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+3nMAssay Description:Inhibition of full length nanoluc-fused FGFR2 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataEC50: 4.26E+3nMAssay Description:Inhibition of full length nanoluc-fused FGFR1 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
Affinity DataIC50: 4.37E+3nMAssay Description:Inhibition of human FGFR1 using poly[Glu:Tyr] (4:1) as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.45E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human FGFR1 using poly[Glu:Tyr] (4:1) as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human wild type FGFR3 using polyEY as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human wild type FGFR3 using polyEY as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human FGFR2 in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 2(Human)
Eberhard Karls University Tubingen
Curated by ChEMBL
Eberhard Karls University Tubingen
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human MAPKAPK2 using KKLNRTLSVA as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 2(Human)
Eberhard Karls University Tubingen
Curated by ChEMBL
Eberhard Karls University Tubingen
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human MAPKAPK2 using KKLNRTLSVA as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human wild type TTK using RBER-CHKtide as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 3(Human)
Eberhard Karls University Tubingen
Curated by ChEMBL
Eberhard Karls University Tubingen
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human MAPKAPK3 using KKLNRTLSVA as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 3(Human)
Eberhard Karls University Tubingen
Curated by ChEMBL
Eberhard Karls University Tubingen
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human MAPKAPK3 using KKLNRTLSVA as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human wild type TTK using RBER-CHKtide as substrate in presence of ATP by hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal GST tagged cytoplasmic domain human FGFR4 (460 to 802 residues) expressed in Escherichia coli BL21 (DE3) using CSox as subst...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of full length nanoluc-fused FGFR1 transfected in HEK293T cells assessed as target engagement incubated for 3 hrs in presence of K10 trace...More data for this Ligand-Target Pair
















