Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50019647
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Cape Town

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 24226BDBM24226(cid_2247 | [3H]-ASTEMIZOLE | Hismanal | ASTEMIZOLE...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human ERG expressed in CHO K1 cells measured after 4 min by QPatch assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Cape Town

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621372BDBM50621372(CHEMBL5434251)
Affinity DataIC50: 420nMAssay Description:Inhibition of human ERG expressed in CHO K1 cells measured after 4 min by QPatch assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Cape Town

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81939BDBM81939(NSC_62969 | VERAPAMIL | CAS_52-53-9)
Affinity DataIC50: 560nMAssay Description:Inhibition of human ERG expressed in CHO K1 cells measured after 4 min by QPatch assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Cape Town

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50609890BDBM50609890(CHEMBL5273140)
Affinity DataIC50: 630nMAssay Description:Inhibition of human ERG expressed in CHO K1 cells measured after 4 min by QPatch assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Cape Town

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621374BDBM50621374(CHEMBL5410878)
Affinity DataIC50: 830nMAssay Description:Inhibition of human ERG expressed in CHO K1 cells measured after 4 min by QPatch assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Cape Town

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621370BDBM50621370(CHEMBL5429029)
Affinity DataIC50: 980nMAssay Description:Inhibition of human ERG expressed in CHO K1 cells measured after 4 min by QPatch assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Cape Town

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621375BDBM50621375(CHEMBL5436114)
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of human ERG expressed in CHO K1 cells measured after 4 min by QPatch assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Cape Town

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621371BDBM50621371(CHEMBL5403581)
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of human ERG expressed in CHO K1 cells measured after 4 min by QPatch assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Cape Town

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50621373BDBM50621373(CHEMBL5434807)
Affinity DataIC50: 5.07E+3nMAssay Description:Inhibition of human ERG expressed in CHO K1 cells measured after 4 min by QPatch assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed