Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50021052
TargetProteasome subunit beta type-9(Human)
Florida International University

Curated by ChEMBL
LigandPNGBDBM50573703(CHEMBL4870740)
Affinity DataIC50: 66nMAssay Description:Inhibition of human LMP2 using Ac-PAL-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 90 min by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProteasome subunit beta type-9(Human)
Florida International University

Curated by ChEMBL
LigandPNGBDBM50573702(CHEMBL4867229)
Affinity DataIC50: 69nMAssay Description:Inhibition of human LMP2 using Ac-PAL-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 90 min by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProteasome subunit beta type-9(Human)
Florida International University

Curated by ChEMBL
LigandPNGBDBM50573704(CHEMBL4855585)
Affinity DataIC50: 87nMAssay Description:Inhibition of human LMP2 using Ac-PAL-AMC as substrate incubated for 1 hr by fluorescence based SpectraMax M5e plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProteasome subunit beta type-9(Human)
Florida International University

Curated by ChEMBL
LigandPNGBDBM50636314(CHEMBL5542874)
Affinity DataIC50: 127nMAssay Description:Inhibition of human LMP2 using Ac-PAL-AMC as substrate incubated for 1 hr by fluorescence based SpectraMax M5e plate readerMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProteasome subunit beta type-9(Human)
Florida International University

Curated by ChEMBL
LigandPNGBDBM50636315(CHEMBL5555733)
Affinity DataIC50: 137nMAssay Description:Inhibition of human LMP2 using Ac-PAL-AMC as substrate incubated for 1 hr by fluorescence based SpectraMax M5e plate readerMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProteasome subunit beta type-9(Human)
Florida International University

Curated by ChEMBL
LigandPNGBDBM50573696(CHEMBL4877277)
Affinity DataIC50: 184nMAssay Description:Inhibition of human LMP2 using Ac-PAL-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 90 min by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProteasome subunit beta type-9(Human)
Florida International University

Curated by ChEMBL
LigandPNGBDBM50636316(CHEMBL5567598)
Affinity DataIC50: 220nMAssay Description:Inhibition of human LMP2 using Ac-PAL-AMC as substrate incubated for 1 hr by fluorescence based SpectraMax M5e plate readerMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProteasome subunit beta type-9(Human)
Florida International University

Curated by ChEMBL
LigandPNGBDBM50573705(CHEMBL4869559)
Affinity DataIC50: 238nMAssay Description:Inhibition of human LMP2 using Ac-PAL-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 90 min by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProteasome subunit beta type-9(Human)
Florida International University

Curated by ChEMBL
LigandPNGBDBM50573707(CHEMBL4866610)
Affinity DataIC50: 262nMAssay Description:Inhibition of human LMP2 using Ac-PAL-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 90 min by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed