Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50021054
Target5-hydroxytryptamine receptor 2A(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50636336(CHEMBL5531940)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]DOI from human 5-HT2AR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 60 mins by scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50636336(CHEMBL5531940)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]DOI from human 5-HT2CR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 60 mins by scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50636336(CHEMBL5531940)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]DOI from human 5-HT2BR expressed in HEK293 cell membrane assessed as inhibition constant incubated for 60 mins by scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50636335(CHEMBL5562096)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]-ketanserin from 5-HT2AR (unknown origin) assessed as inhibition constant by competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed