Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50021784
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644879BDBM50644879(CHEMBL5571548)
Affinity DataKd:  290nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50402023BDBM50402023(BI 6727 | VOLASERTIB)
Affinity DataKd:  900nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644890BDBM50644890(CHEMBL5563717)
Affinity DataKd:  2.03E+3nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644886BDBM50644886(CHEMBL5572400)
Affinity DataKd:  2.15E+3nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644883BDBM50644883(CHEMBL5572259)
Affinity DataKd:  2.79E+3nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644891BDBM50644891(CHEMBL5574577)
Affinity DataKd:  3.95E+3nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644893BDBM50644893(CHEMBL5593934)
Affinity DataKd:  4.24E+3nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644881BDBM50644881(CHEMBL5590858)
Affinity DataKd:  5.26E+3nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644888BDBM50644888(CHEMBL5572922)
Affinity DataKd:  7.36E+3nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644880BDBM50644880(CHEMBL5575481)
Affinity DataKd:  8.06E+3nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644882BDBM50644882(CHEMBL5590594)
Affinity DataKd:  1.42E+4nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644895BDBM50644895(CHEMBL5592268)
Affinity DataKd:  1.54E+4nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644878BDBM50644878(CHEMBL5573507)
Affinity DataKd:  1.68E+4nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644887BDBM50644887(CHEMBL5569873)
Affinity DataKd:  1.68E+4nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644889BDBM50644889(CHEMBL5565607)
Affinity DataKd:  1.73E+4nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644884BDBM50644884(CHEMBL5569336)
Affinity DataKd:  1.75E+4nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644885BDBM50644885(CHEMBL5572333)
Affinity DataKd:  1.92E+4nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644892BDBM50644892(CHEMBL5570042)
Affinity DataKd:  2.01E+4nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644894BDBM50644894(CHEMBL5593133)
Affinity DataKd:  2.09E+4nMAssay Description:Binding affinity to recombinant PLK1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed