Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50021745
Affinity DataIC50: 1.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of PI3Kgamma (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of PI3Kgamma (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 98nMAssay Description:Inhibition of PI3Kdelta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 116nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 129nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 147nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 156nMAssay Description:Inhibition of PI3Kdelta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 157nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 161nMAssay Description:Inhibition of PI3Kdelta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Guizhou Medical University
Curated by ChEMBL
Guizhou Medical University
Curated by ChEMBL
Affinity DataIC50: 162nMAssay Description:Inhibition of PI3Kgamma (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair



























