Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50021750
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 0.960nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of NanoBRET LRRK2 (unknown origin) G2019S mutant expressed in HEK293 cells by NanoBRET TE Intracellular Kinase AssayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 6.70nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 6.70nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of NanoBRET LRRK2 (unknown origin) G2019S mutant expressed in HEK293 cells by NanoBRET TE Intracellular Kinase AssayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Inhibition of NanoBRET LRRK2 (unknown origin) G2019S mutant expressed in HEK293 cells by NanoBRET TE Intracellular Kinase AssayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 8.10nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 8.5nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 9.20nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of NanoBRET LRRK2 (unknown origin) G2019S mutant expressed in HEK293 cells by NanoBRET TE Intracellular Kinase AssayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of wild type human LRRK2 using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human LRRK2 G2019S mutant using [RLGRDKYKTLRQIRQ] peptide substrate by [Gamma33P]-ATP assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of NanoBRET LRRK2 (unknown origin) G2019S mutant expressed in HEK293 cells by NanoBRET TE Intracellular Kinase AssayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of NanoBRET LRRK2 (unknown origin) G2019S mutant expressed in HEK293 cells by NanoBRET TE Intracellular Kinase AssayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 157nMAssay Description:Inhibition of NanoBRET LRRK2 (unknown origin) G2019S mutant expressed in HEK293 cells by NanoBRET TE Intracellular Kinase AssayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Human)
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Korea Advanced Institute of Science and Technology (KAIST)
Curated by ChEMBL
Affinity DataIC50: 333nMAssay Description:Inhibition of NanoBRET LRRK2 (unknown origin) G2019S mutant expressed in HEK293 cells by NanoBRET TE Intracellular Kinase AssayMore data for this Ligand-Target Pair

















