Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50021082
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at CCR6 in C57BL/6J mouse whole blood assessed as inhibition of CCL20-stimulated receptor internalization in lymphocytes incubate...More data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Insurmountable antagonist activity at human CCR6 expressed in HEK293 cells co-transfected with firefly luciferase gene assessed as inhibition of CCL2...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human MDR1More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B3(Human)
Idorsia Pharmaceuticals Ltd.
Curated by ChEMBL
Idorsia Pharmaceuticals Ltd.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of OATP1B3 (unknown origin)More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Human)
Idorsia Pharmaceuticals Ltd.
Curated by ChEMBL
Idorsia Pharmaceuticals Ltd.
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair

