Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50021097
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636720(CHEMBL5558610)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636728(CHEMBL3747105)
Affinity DataEC50:  368nMAssay Description:Agonist activity at alpha9 nAChR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636722(CHEMBL5559353)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636718(CHEMBL5555218)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636718(CHEMBL5555218)
Affinity DataEC50:  510nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636717(CHEMBL5559072)
Affinity DataEC50:  610nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636721(CHEMBL5561644)
Affinity DataEC50:  640nMAssay Description:Partial agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636727(CHEMBL5556786)
Affinity DataEC50:  660nMAssay Description:Agonist activity at alpha9 nAChR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636722(CHEMBL5559353)
Affinity DataEC50:  700nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636719(CHEMBL5517963)
Affinity DataEC50:  830nMAssay Description:Partial agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636727(CHEMBL5556786)
Affinity DataEC50:  980nMAssay Description:Agonist activity at alpha9alpha10 nAChR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636720(CHEMBL5558610)
Affinity DataEC50:  990nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636726(CHEMBL5561901)
Affinity DataEC50:  1.12E+3nMAssay Description:Partial agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636714(CHEMBL3745917)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636716(CHEMBL5532397)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636717(CHEMBL5559072)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636717(CHEMBL5559072)
Affinity DataEC50:  1.30E+3nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636723(CHEMBL5560849)
Affinity DataEC50:  1.49E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636726(CHEMBL5561901)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636719(CHEMBL5517963)
Affinity DataEC50:  1.63E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636722(CHEMBL5559353)
Affinity DataEC50:  1.70E+3nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636723(CHEMBL5560849)
Affinity DataEC50:  2.00E+3nMAssay Description:Partial agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636721(CHEMBL5561644)
Affinity DataEC50:  2.27E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636728(CHEMBL3747105)
Affinity DataEC50:  2.57E+3nMAssay Description:Agonist activity at alpha9alpha10 nAChR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636725(CHEMBL5557858)
Affinity DataEC50:  4.20E+3nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636725(CHEMBL5557858)
Affinity DataEC50:  4.30E+3nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636719(CHEMBL5517963)
Affinity DataEC50:  4.68E+3nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636718(CHEMBL5555218)
Affinity DataEC50:  6.10E+3nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636727(CHEMBL5556786)
Affinity DataEC50:  6.40E+3nMAssay Description:Agonist activity at alpha7 nAChR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636725(CHEMBL5557858)
Affinity DataEC50:  7.00E+3nMAssay Description:Partial agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636715(CHEMBL5568229)
Affinity DataEC50:  9.00E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636715(CHEMBL5568229)
Affinity DataEC50:  1.10E+4nMAssay Description:Partial agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636714(CHEMBL3745917)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636724(CHEMBL5542521)
Affinity DataEC50:  1.50E+4nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636723(CHEMBL5560849)
Affinity DataEC50:  1.80E+4nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636716(CHEMBL5532397)
Affinity DataEC50:  1.80E+4nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM42410(2-acetyloxyethyl(trimethyl)azanium;bromide | MLS00...)
Affinity DataEC50:  2.10E+4nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636716(CHEMBL5532397)
Affinity DataEC50:  2.60E+4nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM42410(2-acetyloxyethyl(trimethyl)azanium;bromide | MLS00...)
Affinity DataEC50:  2.60E+4nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636726(CHEMBL5561901)
Affinity DataEC50:  2.70E+4nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM42410(2-acetyloxyethyl(trimethyl)azanium;bromide | MLS00...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636724(CHEMBL5542521)
Affinity DataEC50:  4.50E+4nMAssay Description:Partial agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636714(CHEMBL3745917)
Affinity DataEC50:  7.60E+4nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636720(CHEMBL5558610)
Affinity DataEC50:  7.83E+4nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636715(CHEMBL5568229)
Affinity DataEC50:  2.80E+5nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50636724(CHEMBL5542521)
Affinity DataEC50:  5.00E+5nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed