Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50021097
Affinity DataEC50: 230nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 368nMAssay Description:Agonist activity at alpha9 nAChR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 480nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Affinity DataEC50: 510nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 610nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 640nMAssay Description:Partial agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured a...More data for this Ligand-Target Pair
Affinity DataEC50: 660nMAssay Description:Agonist activity at alpha9 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 830nMAssay Description:Partial agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured a...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 980nMAssay Description:Agonist activity at alpha9alpha10 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 990nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Affinity DataEC50: 1.12E+3nMAssay Description:Partial agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Affinity DataEC50: 1.15E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 1.18E+3nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Affinity DataEC50: 1.28E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+3nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Affinity DataEC50: 1.49E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Affinity DataEC50: 1.63E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+3nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Partial agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured a...More data for this Ligand-Target Pair
Affinity DataEC50: 2.27E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 2.57E+3nMAssay Description:Agonist activity at alpha9alpha10 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 4.20E+3nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Affinity DataEC50: 4.30E+3nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 4.68E+3nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 6.10E+3nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Affinity DataEC50: 6.40E+3nMAssay Description:Agonist activity at alpha7 nAChR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 7.00E+3nMAssay Description:Partial agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Affinity DataEC50: 9.00E+3nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 1.10E+4nMAssay Description:Partial agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured a...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 1.30E+4nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 1.50E+4nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+4nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+4nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+4nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+4nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+4nMAssay Description:Agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+4nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataEC50: 3.00E+4nMAssay Description:Agonist activity at human alpha9alpha10 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120...More data for this Ligand-Target Pair
Affinity DataEC50: 4.50E+4nMAssay Description:Partial agonist activity at human alpha9 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Affinity DataEC50: 7.60E+4nMAssay Description:Partial agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 12...More data for this Ligand-Target Pair
Affinity DataEC50: 7.83E+4nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+5nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair
Affinity DataEC50: 5.00E+5nMAssay Description:Agonist activity at human alpha7 nAChR expressed as xenopus laevis oocytes assessed as increase in receptor desensitization measured after 120 secs b...More data for this Ligand-Target Pair















