Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50021804
TargetTransient receptor potential cation channel subfamily V member 1(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at capsaicin activated human TRPV1 expressed in HEK293 cells incubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at capsaicin activated human TRPV1 expressed in HEK293 cells incubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 9.71E+3nMAssay Description:Inhibition of human TRPV1 by whole-cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human TRPA1 by whole-cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human TRPV4 by whole-cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 3(Human)
The First Affiliated Hospital of Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50645052(CHEMBL5564691)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human TRPV3 by whole-cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed