Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50021219
Affinity DataKi: 0.600nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of radioligand R-PIA from human adenosine A1 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Displacement of radioligand R-PIA from human adenosine A1 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta scintillation ...More data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Displacement of radioligand R-PIA from human adenosine A1 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Displacement of radioligand R-PIA from human adenosine A1 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Displacement of radioligand I-AB-MECA from human adenosine A3 receptor expressed in CHO cell membrane incubated for 30 mins by microplate beta scinti...More data for this Ligand-Target Pair
Affinity DataKi: 119nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 122nMAssay Description:Displacement of radioligand CGS21680 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta sci...More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membrane incubated for 30 mins by microplate beta scintillation ...More data for this Ligand-Target Pair





























