Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50021962
TargetCoagulation factor X(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50328731(Edoxaban | CHEMBL1269025)
Affinity DataKi:  0.561nMAssay Description:Binding affinity to FXa (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCoagulation factor X(Rat)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM19023(BMS-562247 | CHEMBL231779 | 1-(4-methoxyphenyl)-7-...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to rat FXa assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCoagulation factor X(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM7844(US8822458, 97)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of FXa (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetType-2 angiotensin II receptor(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50646531(Azilsartan medoxomil | Azilsartan medoxomilo | AR-...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of Angiotensin-2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetP2Y purinoceptor 12(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50397205(AR-C126532XX | AZD-6140 | AZD6140 | BRILINTA | TIC...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity to human P2Y12 assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50098320(9-(4-{4-[(4'-Trifluoromethyl-biphenyl-2-carbonyl)-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of MTP (unknown origin) assessed as reduction in triglyceride tranferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetTransthyretin(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50197883(CHEBI:78538 | FX-1006 | Tafamidis | Vyndaqel | US1...)
Affinity DataEC50:  2.70E+3nMAssay Description:Inhibition of wild type human transthyretin extracted from Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProthrombin(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50328731(Edoxaban | CHEMBL1269025)
Affinity DataKi:  6.00E+3nMAssay Description:Binding affinity to thrombin (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50646532(Bempedoic acid | Acide bempedoique | Acido bempedo...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of Acetyl-CoA carboxylase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed