Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50021963
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant human PARL using KSp106 as substrateMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant human PARL using KSp106 as substrateMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant human PARL using KSp106 as substrateMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant human PARL using KSp106 as substrateMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human PARL using KSp106 as substrateMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of recombinant human PARL using KSp106 as substrateMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Inhibition of tetracycline-inducible FLAG-tagged human PARL stably transfected in HEK293T harboring FITR/PARL KOMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human PARL using KSp106 as substrateMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 123nMAssay Description:Inhibition of GlpG in wild-type Escherichia coli MC4100 using MBP-Flag-LacYTMD2-Trx as substrateMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 131nMAssay Description:Inhibition of GlpG in wild-type Escherichia coli MC4100 using MBP-Flag-LacYTMD2-Trx as substrateMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 173nMAssay Description:Inhibition of GlpG in wild-type Escherichia coli MC4100 using MBP-Flag-LacYTMD2-Trx as substrateMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Inhibition of tetracycline-inducible FLAG-tagged human PARL stably transfected in HEK293T harboring FITR/PARL KOMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of Escherichia coli GlpG extracted from Escherichia coli C43(DE3) using KSp96 as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 337nMAssay Description:Inhibition of GlpG in wild-type Escherichia coli MC4100 using MBP-Flag-LacYTMD2-Trx as substrateMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 424nMAssay Description:Inhibition of GlpG in wild-type Escherichia coli MC4100 using MBP-Flag-LacYTMD2-Trx as substrateMore data for this Ligand-Target Pair
TargetPresenilins-associated rhomboid-like protein, mitochondrial(Human)
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 445nMAssay Description:Inhibition of tetracycline-inducible FLAG-tagged human PARL stably transfected in HEK293T harboring FITR/PARL KOMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 1.47E+3nMAssay Description:Inhibition of GlpG in wild-type Escherichia coli MC4100 using MBP-Flag-LacYTMD2-Trx as substrateMore data for this Ligand-Target Pair
TargetRhomboid protease GlpG(Escherichia coli (strain K12))
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science
Curated by ChEMBL
Affinity DataEC50: 1.61E+3nMAssay Description:Inhibition of GlpG in wild-type Escherichia coli MC4100 using MBP-Flag-LacYTMD2-Trx as substrateMore data for this Ligand-Target Pair
