Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50020968
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of PI3Kdelta (unknown origin) using PIP2 as substrate incubated for 2 hrs by TR-FRET analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of PI3Kbeta (unknown origin) using PIP2 as substrate incubated for 2 hrs by TR-FRET analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2 as substrate incubated for 2 hrs by TR-FRET analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of PI3Kgamma (unknown origin) using PIP2 as substrate incubated for 2 hrs by TR-FRET analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Chiesi Farmaceutici S.p.A
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair

