Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50020968
LigandPNGBDBM50323727(2-((9H-purin-6-ylthio)methyl)-5-chloro-3-(2-methox...)
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandPNGBDBM50323727(2-((9H-purin-6-ylthio)methyl)-5-chloro-3-(2-methox...)
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandPNGBDBM50323727(2-((9H-purin-6-ylthio)methyl)-5-chloro-3-(2-methox...)
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandPNGBDBM200639(US9227977, Compound A)
Affinity DataIC50: 12nMAssay Description:Inhibition of PI3Kdelta (unknown origin) using PIP2 as substrate incubated for 2 hrs by TR-FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandPNGBDBM200639(US9227977, Compound A)
Affinity DataIC50: 24nMAssay Description:Inhibition of PI3Kbeta (unknown origin) using PIP2 as substrate incubated for 2 hrs by TR-FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandPNGBDBM200639(US9227977, Compound A)
Affinity DataIC50: 24nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2 as substrate incubated for 2 hrs by TR-FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandPNGBDBM200639(US9227977, Compound A)
Affinity DataIC50: 24nMAssay Description:Inhibition of PI3Kgamma (unknown origin) using PIP2 as substrate incubated for 2 hrs by TR-FRET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
LigandPNGBDBM50323727(2-((9H-purin-6-ylthio)methyl)-5-chloro-3-(2-methox...)
Affinity DataIC50: 180nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed