Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50003811
Affinity DataIC50: 0.110nMAssay Description:Antagonist activity at human P2X7 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of JAK2 (unknown origin) assessed as reduction of EPO-induced STAT5 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of JAK2 (unknown origin) assessed as reduction of EPO-induced STAT5 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Antagonist activity at human P2X7 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Inhibition of p53 (unknown origin) phosphorylation at Ser15 by cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.640nMAssay Description:Inhibition of PI3Kdelta by cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibition of JAK2 (unknown origin) assessed as reduction of EPO-induced STAT5 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of JAK1 (unknown origin) assessed as reduction of IL6-induced STAT3 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Agonist activity at TGR5 in mouse GLUTag cells assessed as secretion of GLP-1 after 2 hrs by HEK293 cell-based luciferase reporter gene assay in pres...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of JAK1 (unknown origin) assessed as reduction of IL6-induced STAT3 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of JAK2 (unknown origin) assessed as reduction of EPO-induced STAT5 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human P2X7 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of PI3Kdelta in neutrophil assessed as inhibition of superoxide production by cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human P2X7 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of JAK2 (unknown origin) assessed as reduction of EPO-induced STAT5 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of JAK2 (unknown origin) assessed as reduction of EPO-induced STAT5 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:Inhibition of JAK2 (unknown origin) assessed as reduction of EPO-induced STAT5 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 235nMAssay Description:Concentration required to inhibit the VCAM-Very late antigen4 (VLA4) interaction in ELISA cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Agonist activity at TGR5 in mouse GLUTag cells assessed as secretion of GLP-1 after 2 hrs by HEK293 cell-based luciferase reporter gene assay in pres...More data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of JAK2 (unknown origin) assessed as reduction of EPO-induced STAT5 phosphorylation by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Agonistic activity in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Concentration required to inhibit the VCAM-Very late antigen4 (VLA4) interaction in ELISA cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Concentration required to inhibit the VCAM-Very late antigen4 (VLA4) interaction in ELISA cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:Concentration required to inhibit the VCAM-Very late antigen4 (VLA4) interaction in ELISA cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 940nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at human P2X7 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Agonistic activity in CHO-hFSHR cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40E+3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20E+3nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Agonistic activity in CHO-hFollicle stimulating hormone receptor cell-based cAMP accumulation assayMore data for this Ligand-Target Pair





























