Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50022122
TargetMu-type opioid receptor(Human)TBA
LigandPNGBDBM50648331(CHEMBL5613639)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to human mu-opioid receptor extracted from CHO cell membrane assessed as inhibition constant incubated for 60 mins in presence of [3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H] U69593 from human kappa-opioid receptor extracted from CHO cell membrane assessed as inhibition constant by liquid scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648330(CHEMBL5611918)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H] U69593 from human kappa-opioid receptor extracted from CHO cell membrane assessed as inhibition constant by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H] DAMGO from rat mu-opioid receptor extracted from CHO cell membrane assessed as inhibition constant by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50207840(H-Tyr-c[pen-Gly-Phe-pen]OH | CHEMBL31421)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H] DPDPE from rat delta-opioid receptor extracted from CHO cell membrane assessed as inhibition constant by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648328(CHEMBL5612630)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H] U69593 from human kappa-opioid receptor extracted from CHO cell membrane assessed as inhibition constant by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648329(CHEMBL5612552)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H] U69593 from human kappa-opioid receptor extracted from CHO cell membrane assessed as inhibition constant by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648328(CHEMBL5612630)
Affinity DataKi:  19nMAssay Description:Displacement of [3H] DAMGO from rat mu-opioid receptor extracted from CHO cell membrane assessed as inhibition constant by liquid scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648331(CHEMBL5613639)
Affinity DataKi:  26nMAssay Description:Binding affinity to human kappa-opioid receptor extracted from CHO cell membrane assessed as inhibition constant incubated for 60 mins in presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648328(CHEMBL5612630)
Affinity DataKi:  201nMAssay Description:Displacement of [3H] DPDPE from rat delta-opioid receptor extracted from CHO cell membrane assessed as inhibition constant by liquid scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed