Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50022186
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50649156(CHEMBL5618354)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human MAGL using 2-arachidonoylglycerol as substrate assessed as reduction in substrate hydrolysis by measuring arachidonic acid format...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50649161(CHEMBL5618586)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of human MAGL using 2-arachidonoylglycerol as substrate assessed as reduction in substrate hydrolysis by measuring arachidonic acid format...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50649160(CHEMBL5620200)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of human MAGL using 2-arachidonoylglycerol as substrate assessed as reduction in substrate hydrolysis by measuring arachidonic acid format...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50649159(CHEMBL5618723)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of human MAGL using 2-arachidonoylglycerol as substrate assessed as reduction in substrate hydrolysis by measuring arachidonic acid format...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50649158(CHEMBL5620312)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of human MAGL using 2-arachidonoylglycerol as substrate assessed as reduction in substrate hydrolysis by measuring arachidonic acid format...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetMonoglyceride lipase(Human)TBA
LigandPNGBDBM50649157(CHEMBL5619084)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of human MAGL using 2-arachidonoylglycerol as substrate assessed as reduction in substrate hydrolysis by measuring arachidonic acid format...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed