Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50021831
Affinity DataKi: 0.600nMAssay Description:Competitive tight binding inhibition of recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence base...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human TMPRSS6 transfected in HEK293SL cells using Boc-QAR-AMC as substrate measured for 24 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Competitive tight binding inhibition of recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence b...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Competitive tight binding inhibition of recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence base...More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Competitive tight binding inhibition of recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence base...More data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.60nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to recombinant human TMPRSS6 using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human Matriptase transfected in HEK293SL cells using Boc-QAR-AMC as substrate measured for 24 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human TMPRSS6 transfected in HEK293SL cells using Boc-QAR-AMC as substrate measured for 24 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of recombinant human thrombin using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Binding affinity to recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Mixed inhibition of recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of recombinant human thrombin using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 323nMAssay Description:Inhibition of FXA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 332nMAssay Description:Inhibition of human TMPRSS6 transfected in HEK293SL cells using Boc-QAR-AMC as substrate measured for 24 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 352nMAssay Description:Inhibition of human Matriptase transfected in HEK293SL cells using Boc-QAR-AMC as substrate measured for 24 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 395nMAssay Description:Inhibition of recombinant human thrombin using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 618nMAssay Description:Mixed inhibition of recombinant human Matriptase using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.32E+3nMAssay Description:Inhibition of recombinant human FXA using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6.07E+3nMAssay Description:Inhibition of human Matriptase transfected in HEK293SL cells using Boc-QAR-AMC as substrate measured for 24 hrsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human furin using Boc-RVRR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human furin using Boc-RVRR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human furin using Boc-RVRR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human FXA using Boc-QAR-AMC as substrate assessed as inhibition constant by fluorescence based analysisMore data for this Ligand-Target Pair














