Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50022061
TargetSodium channel protein type 2 subunit alpha(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50647649(CHEMBL5598329)
Affinity DataIC50: 65nMAssay Description:Inhibition of human Nav1.2 expressed in HEK293 cells at -40 mv holding potential measured after 5 mins by whole cell voltage clamp electrophysiologic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50647647(CHEMBL5598304)
Affinity DataIC50: 120nMAssay Description:Inhibition of human Nav1.2 expressed in HEK293 cells at -40 mv holding potential measured after 5 mins by whole cell voltage clamp electrophysiologic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50647649(CHEMBL5598329)
Affinity DataIC50: 158nMAssay Description:Inhibition of human Nav1.2 expressed in HEK293 cells at -120 mv holding potential measured after 5 mins by whole cell voltage clamp electrophysiologi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50647651(CHEMBL5596160)
Affinity DataIC50: 180nMAssay Description:Inhibition of Nav1.2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50647648(CHEMBL5598220)
Affinity DataIC50: 635nMAssay Description:Inhibition of human Nav1.2 expressed in HEK293 cells at -40 mv holding potential measured after 5 mins by whole cell voltage clamp electrophysiologic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50647650(Elpetrigine | Elpetrigina | JZP-4)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Nav1.2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50647647(CHEMBL5598304)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human Nav1.2 expressed in HEK293 cells at -120 mv holding potential measured after 5 mins by whole cell voltage clamp electrophysiologi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50647648(CHEMBL5598220)
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of human Nav1.2 expressed in HEK293 cells at -120 mv holding potential measured after 5 mins by whole cell voltage clamp electrophysiologi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed