Compile Data Set for Download or QSAR
Report error Found 93 Enz. Inhib. hit(s) with all data for entry = 50021907
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646035(CHEMBL5591488)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646005(CHEMBL5591695)
Affinity DataIC50: 0.430nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646015(CHEMBL5593700)
Affinity DataIC50: 0.720nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646030(CHEMBL5594475)
Affinity DataIC50: 0.850nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646014(CHEMBL5591879)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646029(CHEMBL5592778)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646016(CHEMBL5594221)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646040(CHEMBL5592978)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646040(CHEMBL5592978)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of full length N-terminal his-tagged human OGA expressed in baculovirus expression system preincubated for for 30 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646041(Ly-3372689 | LY3372689 | Ceperognastat)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of full length N-terminal his-tagged human OGA expressed in baculovirus expression system preincubated for for 30 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646036(CHEMBL5590780)
Affinity DataIC50: 3nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646039(CHEMBL5593511)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50645993(CHEMBL5579695)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646009(CHEMBL5592385)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646006(CHEMBL5591089)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50645988(CHEMBL5591704)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646034(CHEMBL5591551)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646033(CHEMBL5591513)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50645987(CHEMBL5583946)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646038(CHEMBL5584048)
Affinity DataEC50:  6.90nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646033(CHEMBL5591513)
Affinity DataEC50:  7.5nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646027(CHEMBL5591099)
Affinity DataIC50: 8nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646010(CHEMBL5591460)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50645994(CHEMBL5595991)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646038(CHEMBL5584048)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646026(CHEMBL5591200)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646024(CHEMBL5590193)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM508589(US11046712, No 69)
Affinity DataIC50: 10nMAssay Description:Inhibition of human OGAMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646012(CHEMBL5591950)
Affinity DataIC50: 10nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646037(CHEMBL5592023)
Affinity DataEC50:  11nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646004(CHEMBL5594139)
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646037(CHEMBL5592023)
Affinity DataIC50: 12nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646039(CHEMBL5593511)
Affinity DataEC50:  13nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646023(CHEMBL5592284)
Affinity DataIC50: 16nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646017(CHEMBL5595937)
Affinity DataIC50: 16nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50645990(CHEMBL5592814)
Affinity DataIC50: 19nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646004(CHEMBL5594139)
Affinity DataEC50:  21nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50323697(thiamet-G | (3AR,5R,6S,7R,7AR)-2-(ETHYLAMINO)-5-(H...)
Affinity DataKi:  21nMAssay Description:Binding affinity to human O-GlcNAcase assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50645985(CHEMBL5593028)
Affinity DataIC50: 23nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646040(CHEMBL5592978)
Affinity DataEC50:  23nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646008(CHEMBL5591919)
Affinity DataIC50: 24nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646028(CHEMBL5592529)
Affinity DataIC50: 24nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646027(CHEMBL5591099)
Affinity DataEC50:  25nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646020(CHEMBL5593505)
Affinity DataIC50: 25nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646021(CHEMBL5590863)
Affinity DataIC50: 26nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646014(CHEMBL5591879)
Affinity DataEC50:  26nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646035(CHEMBL5591488)
Affinity DataEC50:  28nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50646025(CHEMBL5595069)
Affinity DataIC50: 29nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Human)TBA
LigandPNGBDBM50645992(CHEMBL5590741)
Affinity DataIC50: 32nMAssay Description:Inhibition of GST-tagged human recombinant OGA using fuoresceinmono-beta-o-N-acetylglucosarnine as substrate incubated for 60 mins under dark conditi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtein O-GlcNAcase(Rat)TBA
LigandPNGBDBM50646028(CHEMBL5592529)
Affinity DataEC50:  32nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
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