Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50023448
Affinity DataIC50: 0.75nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.890nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.30nMAssay Description:Inhibition of EGFR L858R/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.40nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.60nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.70nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.10nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.40nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.5nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.60nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.70nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.80nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.60nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 3.70nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 5.10nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6.80nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 8.5nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 9.70nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 9.80nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 11nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 13nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 13nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 14nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 20nMAssay Description:Inhibition of EGFR de119/T790M/C797S mutant (694 to 1022 residues)(unknown origin) using BML-P243 as substrate incubated for 90 mins in presence of A...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 21nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 22nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 24nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 45nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 66nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 215nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 237nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 275nMAssay Description:Inhibition of N-terminal GST-tagged wild-type human EGFR (669 to 1210 residues) expressed in Sf21 cells using BML-P243 as substrate incubated for 90 ...More data for this Ligand-Target Pair
Ligand Info
